Bupranololum

Bupranololum Uses, Dosage, Side Effects, Food Interaction and all others data.

Bupranololum is a non-selective beta blocker with potency similar to propanolol. It does not have intrinsic sympathomimetic activity (ISA), but does have strong membrane stabilizing activity.

Bupranololum is a competitive, nonselective beta-blocker similar to propanolol without intrinsic sympathomimetic activity.

Trade Name Bupranololum
Generic Bupranolol
Bupranolol Other Names Bupranolol, Bupranololum
Type
Formula C14H22ClNO2
Weight Average: 271.783
Monoisotopic: 271.13390666
Protein binding

76%

Groups Experimental
Therapeutic Class
Manufacturer
Available Country
Last Updated: September 19, 2023 at 7:00 am
Bupranololum
Bupranololum

Uses

Used to manage hypertension and tachycardia. Also used to treat glaucoma.

How Bupranololum works

Bupranololum competes with sympathomimetic neurotransmitters such as catecholamines for binding at beta(1)-adrenergic receptors in the heart, inhibiting sympathetic stimulation. This results in a reduction in resting heart rate, cardiac output, systolic and diastolic blood pressure, and reflex orthostatic hypotension.

Toxicity

Symptoms of overdose include bradycardia, cardiac failure, hypotension, and brochospasm.

Elimination Route

Quickly and completely absorbed from the gut with less than 10% oral bioavailability.

Half Life

2-4 hours

Innovators Monograph

You find simplified version here Bupranololum

*** Taking medicines without doctor's advice can cause long-term problems.
Share